e-Article
Identification and Optimization of a Ligand-Efficient Benzoazepinone Bromodomain and Extra Terminal (BET) Family Acetyl-Lysine Mimetic into the Oral Candidate Quality Molecule I-BET432
Document Type
Article
Author
Humphreys, P.G.; Anderson, N.A.; Bamborough, P.; Baxter, A.; Chung, C.-W.; Cookson, R.; Craggs, P.D.; Dalton, T.; Fournier, J.C.L.; Gordon, L.J.; Gray, H.F.; Gray, M.W.; Gregory, R.; Hirst, D.J.; Jones, K.L.; Kessedjian, H.; Lugo, D.; McGonagle, G.; Patel, V.K.; Patten, C.; Poole, D.L.; Prinjha, R.K.; Ramirez-Molina, C.; Rioja, I.; Seal, G.; Stafford, K.A.J.; Shah, R.R.; Tape, D.; Theodoulou, N.H.; Tomlinson, L.; Ukuser, S.; Wall, I.D.; Wellaway, N.; White, G.; Jamieson, C.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 24 November 2022, 65(22):15174-15207)
Subject
Language
English
ISSN
15204804
00222623
00222623