학술논문
Discovery of AZD4573, a Potent and Selective Inhibitor of CDK9 That Enables Short Duration of Target Engagement for the Treatment of Hematological Malignancies
Document Type
Article
Author
Barlaam, B.; Dishington, A.; Donald, C.S.; Glossop, S.; Hawkins, J.; Holmes, J.; McGuire, T.M.; Moore, J.E.; Pike, A.; Pike, K.G.; Roberts, B.; Stead, D.; Sumner, N.; Casella, R.; Wang, J.; Wu, D.; Cidado, J.; De Savi, C.; Drew, L.; Ferguson, D.; Grebe, T.; Gu, C.; Hande, S.; Hird, A.W.; Horstick, J.; Lamb, M.L.; Proia, T.; San Martin, M.; Sarkar, U.; Shao, W.; Thakur, K.; Vasbinder, M.M.; Varnes, J.G.; Yang, B.; Cook, C.; Ferguson, A.D.; O'Connell, N.; Jiang, Y.; Wang, L.; Wu, L.; Yao, T.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 24 December 2020, 63(24):15564-15590)
Subject
Language
English
ISSN
15204804
00222623
00222623