학술논문
Structure-Based Design and Preclinical Characterization of Selective and Orally Bioavailable Factor XIa Inhibitors: Demonstrating the Power of an Integrated S1 Protease Family Approach
Document Type
Article
Author
Roache, J.; Barnes-Seeman, D.; Turner, G.; Duvadie, R.; Hornak, V.; Karki, R.G.; Weihofen, W.A.; Calhoun, A.; Fazal, T.; Liu, D.; Kirman, L.; Bevan, D.; Mo, R.; Zessis, R.; Huang, X.; Lindsley, L.; Currie, T.; Chiu, Y.-H.; Fridrich, C.; Delgado, P.; Wang, S.; Hollis-Symynkywicz, M.; Williams, E.; Liu, H.; Liang, G.; Kim, H.; Hoffmann, P.; Elliott, J.; Adams, C.M.; Lorthiois, E.; Altmann, E.; Hassiepen, U.; Schiering, N.; Perruccio, F.; Dedic, D.; Durand, C.; Dussauge, S.; Fettis, K.; Tritsch, F.; Dentel, C.; Druet, A.; Lachal, J.; Namoto, K.; Monnet, G.; Muller, L.; Berghausen, J.; Hein, A.; Ramage, P.; D'arcy, A.; Harlfinger, S.; Renatus, M.; Ruedisser, S.; Sedrani, R.; Maibaum, J.; Feldman, D.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 13 August 2020, 63(15):8088-8113)
Subject
Language
English
ISSN
15204804
00222623
00222623