학술논문
Identification of N-{cis-3-[Methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune Diseases
Document Type
Article
Author
Vazquez, M.L.; Kaila, N.; Strohbach, J.W.; Trzupek, J.D.; Unwalla, R.; Brown, M.F.; Flanagan, M.E.; Mitton-Fry, M.J.; Arnold, E.P.; Basak, A.; Heasley, S.E.; Kwon, S.; Langille, J.; Parikh, M.D.; Casavant, J.M.; Harris, T.M.; Han, S.; Caspers, N.; Yang, X.; Banker, M.E.; Robinson, R.P.; Griffin, S.H.; Dowty, M.E.; Hegen, M.; Symanowicz, P.T.; Li, L.; Wang, L.; Lin, T.H.; Jussif, J.; Clark, J.D.; Telliez, J.-B.; Johnson, T.A.; Duclos, B.A.; Fenwick, A.E.; Tenbrink, R.E.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 8 February 2018, 61(3):1130-1152)
Subject
Language
English
ISSN
15204804
00222623
00222623