학술논문
Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit
Document Type
Article
Author
Gerstenberger, B.S.; Trzupek, J.D.; Bunnage, M.E.; Owen, D.R.; Tallant, C.; Fedorov, O.; Filippakopoulos, P.; Brennan, P.E.; Fedele, V.; Martin, S.; Picaud, S.; Rogers, C.; Müller, S.; Knapp, S.; Parikh, M.; Taylor, A.; Samas, B.; O'Mahony, A.; Berg, E.; Pallares, G.; Torrey, A.D.; Treiber, D.K.; Samardjiev, I.J.; Nasipak, B.T.; Padilla-Benavides, T.; Wu, Q.; Imbalzano, A.N.; Nickerson, J.A.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 26 May 2016, 59(10):4800-4811)
Subject
Language
English
ISSN
15204804
00222623
00222623