학술논문
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Academic Journal
Brousseau, M.E.; Clairmont, K.B.; Flyer, A.N.; Golosov, A.A.; Amin, J.; Burdick, D.; Caplan, S.; Chen, G.; Chopra, R.; Ames, L.; Dubiel, D.; Fan, L.; Kelly-Sullivan, D.; Koch, A.W.; Li, J.; Liu, E.; Lubicka, D.; Nakajima, K.; Nettleton, D.; Pan, M.; Patel, T.; Perry, L.; Poirier, J.; Seepersaud, M.; Subramanian, V.; Vera, V.; Xu, M.; Yang, L.; Yang, Q.; Yu, J.; Zhu, G.; Monovich, L.G.; Spraggon, G.; Grosche, P.; Andre, J.; Gattlen, R.; Lewis, I.; Marzinzik, A.; Ottl, J.; Pickett, S.; Pelle, X.; Reid, P.C.
In: Cell Chemical Biology . (Cell Chemical Biology, 17 February 2022, 29(2):249-258.e5)
Academic Journal
In: ACS Combinatorial Science . (ACS Combinatorial Science, 9 March 2020, 22(3):120-128)
Discovery of Asciminib (ABL001), an Allosteric Inhibitor of the Tyrosine Kinase Activity of BCR-ABL1
Academic Journal
Schoepfer, J.; Jahnke, W.; Cotesta, S.; Cowan-Jacob, S.W.; Drueckes, P.; Gabriel, T.; Groell, J.-M.; Grotzfeld, R.M.; Henry, C.; Jones, D.; Manley, P.W.; Pellé, X.; Rummel, G.; Salem, B.; Zoller, T.; Marzinzik, A.L.; Furet, P.; Dodd, S.; Loo, A.; Berellini, G.; Buonamici, S.; Fabbro, D.; Hassan, A.Q.; Iyer, V.; Lombardo, F.; Warmuth, M.; Wylie, A.A.
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 27 September 2018, 61(18):8120-8135)
Academic Journal
Wylie, A.A.; Loo, A.; Donovan, J.; Zhu, W.; Buonamici, S.; Hassan, A.Q.; Lombardo, F.; Palmer, M.; Berellini, G.; Dodd, S.; Thohan, S.; Bitter, H.; Petruzzelli, L.; Vanasse, K.G.; Warmuth, M.; Keen, N.J.; Sellers, W.R.; Schoepfer, J.; Jahnke, W.; Cowan-Jacob, S.W.; Furet, P.; Marzinzik, A.L.; Pelle, X.; Iyer, V.; Hofmann, F.; Branford, S.; Ross, D.M.; Hughes, T.P.
In: Nature . (Nature, 30 March 2017, 543(7647):733-737)
Academic Journal
Jahnke, W.; Bold, G.; Marzinzik, A.L.; Ofner, S.; Pellé, X.; Cotesta, S.; Bourgier, E.; Lehmann, S.; Henry, C.; Hemmig, R.; Stauffer, F.; Hartwieg, J.C.D.; Green, J.R.; Rondeau, J.-M.
In: Angewandte Chemie - International Edition . (Angewandte Chemie - International Edition, 23 November 2015, 54(48):14575-14579)
Academic Journal
Marzinzik, A.L.; Amstutz, R.; Bold, G.; Bourgier, E.; Cotesta, S.; Glickman, J.F.; Götte, M.; Henry, C.; Lehmann, S.; Hartwieg, J.C.D.; Ofner, S.; Pellé, X.; Roddy, T.P.; Rondeau, J.-M.; Stauffer, F.; Stout, S.J.; Widmer, A.; Zimmermann, J.; Zoller, T.; Jahnke, W.
In: ChemMedChem . (ChemMedChem, 1 November 2015, 10(11):1884-1891)
Academic Journal
Jahnke, W.; Grotzfeld, R.M.; Pellé, X.; Strauss, A.; Fendrich, G.; Cowan-Jacob, S.W.; Cotesta, S.; Fabbro, D.; Furet, P.; Mestan, J.; Marzinzik, A.L.
In: Journal of the American Chemical Society . (Journal of the American Chemical Society, 26 May 2010, 132(20):7043-7048)
Academic Journal
Fabbro, D.; Manley, P.W.; Jahnke, W.; Liebetanz, J.; Szyttenholm, A.; Fendrich, G.; Strauss, A.; Warmuth, M.; Pelle, X.; Grotzfeld, R.; Berst, F.; Marzinzik, A.; Cowan-Jacob, S.W.; Furet, P.; Mestan, J.; Adrian, F.; Zhang, J.; Gray, N.S.
In: Biochimica et Biophysica Acta - Proteins and Proteomics . (Biochimica et Biophysica Acta - Proteins and Proteomics, March 2010, 1804(3):454-462)
Academic Journal
Jahnke, W.; Rondeau, J.-M.; Cotesta, S.; Marzinzik, A.; Pellé, X.; Geiser, M.; Strauss, A.; Götte, M.; Bitsch, F.; Hemmig, R.; Henry, C.; Lehmann, S.; Glickman, J.F.; Roddy, T.P.; Stout, S.J.; Green, J.R.
In: Nature Chemical Biology . (Nature Chemical Biology, September 2010, 6(9):660-666)
Academic Journal
In: Synlett . (Synlett, 4 October 2005, (16):2441-2444)
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[AR] Pellé, X.
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