학술논문
Discovery and Clinical Proof-of-Concept of RLY-2608, a First-in-Class Mutant-Selective Allosteric PI3Kalpha Inhibitor That Decouples Antitumor Activity from Hyperinsulinemia
Document Type
Journal
Author
Varkaris, Andreas; Pazolli, Ermira; Gunaydin, Hakan; Wang, Qi; Pierce, Levi; Boezio, Alessandro A.; Bulku, Artemisa; Dipietro, Lucian; Fridrich, Cary; Frost, Adam; Giordanetto, Fabrizio; Hamilton, Erika P.; Harris, Katherine; Holliday, Michael; Hunter, Tamieka L.; Iskandar, Amanda; Ji, Yongli; Larivee, Alexandre; Larochelle, Jonathan R.; Lescarbeau, Andre; Llambi, Fabien; Lormil, Brenda; Mader, Mary M.; Mar, Brenton G.; Martin, Iain; Mclean, Thomas H.; Michelsen, Klaus; Pechersky, Yakov; Puente-Poushnejad, Erika; Raynor, Kevin; Rogala, Dipali; Samadani, Ramin; Schram, Alison M.; Shortsleeves, Kelley; Swaminathan, Sweta; Tajmir, Shahein; Tan, Gege; Tang, Yong; Valverde, Roberto; Wehrenberg, Bryan; Wilbur, Jeremy; Williams, Bret R.; Zeng, Hongtao; Zhang, Hanmo; Walters, W. Patrick; Wolf, Beni B.; Shaw, David E.; Bergstrom, Donald A.; Watters, James; Fraser, James S.; Fortin, Pascal D.; Kipp, D. Randal
Source
Subject
Language
English
ISSN
21598290