학술논문
(3R,5S,E)-7-(4-(4-fluorophenyl)-6-isopropyl-2-(methyl(1-methyl-1H-1,2,4-triazo1-5-yl)amino)pyrimidin-5-yl)-3,5-dihydroxyhept-6-enoic acid (BMS-644950): A rationally designed orally efficacious 3-hydroxy-3-methylglutaryl coenzyme-A reductase inhibitor with reduced myotoxicity potential
Document Type
Journal
Author
Ahmad, Saleem; Madsen, Cort S.; Stein, Philip D.; Janovitz, Evan; Huang, Christine; Ngu, Khehyong; Bisaha, Sharon; Kennedy, Lawrence J.; Chen, Bang-Chi; Zhao, Rulin; Sitkoff, Doree; Monshizadegan, Hossain; Yin, Xiaohong; Ryan, Carol S.; Zhang, Rongan; Giancarli, Mary; Bird, Eileen; Chang, Ming; Chen, Xing; Setters, Robert; Search, Debra; Zhuang, Shaobin; Nguyen-Tran, Van; Cuff, Carolyn A.; Harrity, Thomas; Darienzo, Celia J.; Li, Tong; Reeves, Richard A.; Blanar, Michael A.; Barrish, Joel C.; Zahler, Robert; Robl, Jeffrey A.
Source
Subject
Language
English
ISSN
00222623