학술논문
Discovery of (1S,2R,3S,4S,5R,6R)-2-Amino-3-[(3,4-difluorophenyl)sulfanylmethyl]-4-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid Hydrochloride (LY3020371·HCl): A Potent, Metabotropic Glutamate 2/3 Receptor Antagonist with Antidepressant-Like Activity
Document Type
Article
Author
Chappell, M.D.; Li, R.; Smith, S.C.; Dressman, B.A.; Tromiczak, E.G.; Tripp, A.E.; Blanco, M.-J.; Vetman, T.; Quimby, S.J.; Matt, J.; Britton, T.C.; Fivush, A.M.; Schkeryantz, J.M.; Mayhugh, D.; Erickson, J.A.; Bures, M.G.; Monn, J.A.; Mitch, C.H.; Ornstein, P.L.; Wang, X.-S.; Heinz, B.A.; Jaramillo, C.; Carpintero, M.; Diego, J.E.D.; Barberis, M.; Garcia-Cerrada, S.; Soriano, J.F.; Antonysamy, S.; Atwell, S.; Macewan, I.; Condon, B.; Sougias, C.; Wang, J.; Zhang, A.; Conners, K.; Groshong, C.; Wasserman, S.R.; Koss, J.W.; Wafford, K.A.; Seidel, W.; Swanson, S.; Catlow, J.T.; Bedwell, D.W.; Witkin, J.M.; Li, X.; Overshiner, C.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 22 December 2016, 59(24):10974-10993)
Subject
Language
English
ISSN
15204804
00222623
00222623