학술논문
Driving Potency with Rotationally Stable Atropisomers: Discovery of Pyridopyrimidinedione-Carbazole Inhibitors of BTK
Document Type
Article
Author
Srivastava, A.S.; Ko, S.; Watterson, S.H.; Pattoli, M.A.; Skala, S.; Cheng, L.; Obermeier, M.T.; Vickery, R.; Discenza, L.N.; D'Arienzo, C.J.; Gillooly, K.M.; Taylor, T.L.; Pulicicchio, C.; McIntyre, K.W.; Yip, S.; Li, P.; Sun, D.; Wu, D.-R.; Dai, J.; Wang, C.; Zhang, Y.; Wang, B.; Pawluczyk, J.; Kempson, J.; Zhao, R.; Hou, X.; Rampulla, R.; Mathur, A.; Galella, M.A.; Salter-Cid, L.; Barrish, J.C.; Carter, P.H.; Fura, A.; Burke, J.R.; Tino, J.A.
Source
In: ACS Medicinal Chemistry Letters . (ACS Medicinal Chemistry Letters, 12 November 2020, 11(11):2195-2203)
Subject
Language
English
ISSN
19485875