학술논문
Discovery of 5-chloro-4-((1-(5-chloropyrimidin-2-yl)piperidin-4-yl)oxy)-1-(2-fluoro-4-(methylsulfonyl)phenyl)pyridin-2(1 H)-one (BMS-903452), an antidiabetic clinical candidate targeting GPR119
Document Type
Article
Author
Wacker, D.A.; Wang, Y.; Broekema, M.; Rossi, K.; Oconnor, S.; Hong, Z.; Wu, G.; Malmstrom, S.E.; Hung, C.-P.; Lamarre, L.; Chimalakonda, A.; Zhang, L.; Xin, L.; Cai, H.; Chu, C.; Boehm, S.; Zalaznick, J.; Ponticiello, R.; Sereda, L.; Han, S.-P.; Zebo, R.; Zinker, B.; Luk, C.E.; Wong, R.; Everlof, G.; Li, Y.-X.; Wu, C.K.; Lee, M.; Griffen, S.; Miller, K.J.; Krupinski, J.; Robl, J.A.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 25 September 2014, 57(18):7499-7508)
Subject
Language
English
ISSN
15204804
00222623
00222623