학술논문
Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design
Document Type
Article
Author
Gavai, A.V.; Norris, D.; Delucca, G.; Tortolani, D.; Tokarski, J.S.; Dodd, D.; O'Malley, D.; Zhao, Y.; Quesnelle, C.; Gill, P.; Vaccaro, W.; Huynh, T.; Ahuja, V.; Han, W.-C.; Mussari, C.; Harikrishnan, L.; Kamau, M.; Poss, M.; Sheriff, S.; Yan, C.; Marsilio, F.; Menard, K.; Wen, M.-L.; Rampulla, R.; Wu, D.-R.; Li, J.; Zhang, H.; Li, P.; Sun, D.; Yip, H.; Traeger, S.C.; Zhang, Y.; Mathur, A.; Zhang, H.; Huang, C.; Yang, Z.; Ranasinghe, A.; Everlof, G.; Raghavan, N.; Tye, C.K.; Wee, S.; Hunt, J.T.; Vite, G.; Westhouse, R.; Lee, F.Y.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 14 October 2021, 64(19):14247-14265)
Subject
Language
English
ISSN
15204804
00222623
00222623