학술논문
The Identification of Potent, Selective, and Orally Available Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase: The Discovery of AZD0156 (8-{6-[3-(Dimethylamino)propoxy]pyridin-3-yl}-3-methyl-1-(tetrahydro-2 H-pyran-4-yl)-1,3-dihydro-2 H-imidazo[4,5- c]quinolin-2-one)
Document Type
Article
Author
Pike, K.G.; Barlaam, B.; Cadogan, E.; Colclough, N.; Davies, N.L.; De-Almeida, C.; Degorce, S.L.; Durant, S.T.; Hughes, G.D.; McGuire, T.M.; Pass, M.; Robb, G.; Wilson, J.; Campbell, A.; Chen, Y.; Al-Huniti, N.; Dishington, A.; Hassall, L.A.; Holmes, J.; Macfaul, P.A.; Mulholland, K.R.; Didelot, M.; Ducray, R.; Ouvry, G.; Stratton, N.; Wang, Z.; Zhai, B.; Zhao, K.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 10 May 2018, 61(9):3823-3841)
Subject
Language
English
ISSN
15204804
00222623
00222623