학술논문
Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle
Document Type
Article
Author
Mackman, R.L.; Jansa, P.; Appleby, T.; Cai, R.; Cannizzaro, C.; Chin, G.; Hui, H.; Ji, M.; Jin, H.; Karki, K.; Lee, Y.-J.; Liclican, A.; Mish, M.; Murray, B.; Pyun, P.; Sangi, M.; Santos, R.; Schmitz, U.; Schrier, A.; Siegel, D.; Sperandio, D.; Stepan, G.; Tian, Y.; Yang, H.; Schultz, B.E.; Steadman, V.A.; Dean, D.K.; Poullennec, K.G.; Austin, C.; Blakemore, C.A.; Chiva, J.-Y.C.; Dunbar, N.A.; Highton, A.J.; Keats, A.J.; Lazarides, L.; Pettit, S.B.; Sanvoisin, J.; Watt, G.M.; Fliri, H.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 8 November 2018, 61(21):9473-9499)
Subject
Language
English
ISSN
15204804
00222623
00222623