학술논문
Discovery of a thiadiazole-pyridazine-based allosteric glutaminase 1 inhibitor series that demonstrates oral bioavailability and activity in tumor xenograft models
Document Type
Article
Author
Finlay, M.R.V.; Anderton, M.; Bailey, A.; Boyd, S.; Critchlow, S.E.; Culshaw, J.; Hollingsworth, I.; Littleson, M.; Mooney, L.; Nissink, J.W.M.; Perkins, D.; Powell, S.; Raubo, P.; Smith, P.D.; Stark, A.; Ting, A.; Wilson, Z.; Winter-Holt, J.J.; Wood, J.M.; Wrigley, G.L.; Brookfield, J.; Cairnduff, C.; Charles, M.; Cheasty, A.; Ekwuru, T.; Jones, N.; Leroux, F.; McCarron, H.; McKelvie, J.; Quesada, M.J.; Sabin, V.; Smith, J.; Wang, P.; Yu, G.; Zhang, P.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 25 July 2019, 62(14):6540-6560)
Subject
Language
English
ISSN
15204804
00222623
00222623