학술논문
Rationally Designed, Conformationally Constrained Inverse Agonists of RORγt - Identification of a Potent, Selective Series with Biologic-Like in Vivo Efficacy
Document Type
Article
Author
Marcoux, D.; Duan, J.J.-W.; Shi, Q.; Cherney, R.J.; Srivastava, A.S.; Cornelius, L.; Batt, D.G.; Liu, Q.; Beaudoin-Bertrand, M.; Weigelt, C.A.; Khandelwal, P.; Rampulla, R.A.; Mathur, A.; Yip, S.; Li, P.; Wu, D.-R.; Khan, J.; Ruzanov, M.; Sack, J.S.; Wang, J.; Yarde, M.; Cvijic, M.E.; Li, S.; Shuster, D.J.; Borowski, V.; Xie, J.H.; Mcintyre, K.W.; Obermeier, M.T.; Fura, A.; Stefanski, K.; Cornelius, G.; Hynes, J.; Tino, J.A.; Macor, J.E.; Salter-Cid, L.; Denton, R.; Zhao, Q.; Carter, P.H.; Dhar, T.G.M.; Vishwakrishnan, S.; Selvakumar, K.; Karmakar, A.; Gupta, A.K.; Basha, M.; Ramlingam, S.; Manjunath, N.; Vanteru, S.; Karmakar, S.; Maddala, N.; Vetrichelvan, M.; Gupta, A.
Source
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 14 November 2019, 62(21):9931-9946)
Subject
Language
English
ISSN
15204804
00222623
00222623