학술논문
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Academic Journal
Dzierba, C.D.; Bronson, J.J.; Dasgupta, B.; Karageorge, G.; Macor, J.E.; Kostich, W.; Easton, A.; Bourin, C.; Westphal, R.; Bristow, L.J.; Conway, C.M.; Hamman, B.; Allen, J.; Esposito, K.M.; Padmanabha, R.; Lippy, J.S.; Grace, J.; Lentz, K.; Morrison, J.; Morgan, D.; Browning, M.R.; Parker, D.D.; Santone, K.S.; Rajamani, R.; Good, A.; Muckelbauer, J.K.; Khan, J.; Camac, D.; Ghosh, K.; Halan, V.; Denton, R.R.
In: Medicinal Chemistry Research . (Medicinal Chemistry Research, July 2023, 32(7):1369-1375)
Academic Journal
Regueiro-Ren, A.; Meanwell, N.A.; Sit, S.-Y.; Chen, Y.; Chen, J.; Swidorski, J.J.; Liu, Z.; Venables, B.L.; Sin, N.; Hartz, R.A.; Protack, T.; Lin, Z.; Zhang, S.; Li, Z.; Cockett, M.; Dicker, I.; Krystal, M.; Wu, D.-R.; Li, P.; Kempson, J.; Hou, X.; Rampulla, R.; Mathur, A.; Gupta, A.; Park, H.; Sarjeant, A.; Benitex, Y.; Rahematpura, S.; Parker, D.; Phillips, T.; Haskell, R.; Jenkins, S.; Santone, K.S.; Hanumegowda, U.
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 22 September 2022, 65(18):11927-11948)
Academic Journal
Luo, G.; Chen, L.; Ditta, J.; Bronson, J.J.; MacOr, J.E.; Dzierba, C.D.; Kostich, W.A.; Easton, A.; Bourin, C.; Gulianello, M.; Conway, C.M.; Li, Y.-W.; Pieschl, R.; Tian, Y.; Hong, Y.; Bristow, L.; Albright, C.F.; Hamman, B.; Allen, J.; Wilson, A.; Gopinathan, S.; Wason, S.; Lippy, J.; Nara, S.; Maishal, T.K.; Thiyagarajan, K.; Jalagam, P.; Pattipati, S.N.; Dandapani, K.; Dokania, M.; Vattikundala, P.; Sharma, V.; Elavazhagan, S.; Verma, M.K.; Das, M.L.; Wagh, S.; Saminathan, H.; Holenarsipur, V.K.; Kumar, A.; Rao, A.; Putlur, S.P.; Sarvasiddhi, S.K.; Shankar, G.; Louis, J.V.; Ramarao, M.; Vetrichelvan, M.; Gupta, A.; Balakrishnan, A.; Johnson, B.M.; Santone, K.S.; Thalody, G.; Denton, R.; Mathur, A.; Li, J.; Smith, D.; Pawluczyk, J.; Sun, D.; Yip, S.; Wu, D.-R.
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 24 March 2022, 65(6):4457-4480)
Academic Journal
Luo, G.; Chen, L.; Bronson, J.J.; MacOr, J.E.; Dzierba, C.D.; Kostich, W.A.; Easton, A.; Bourin, C.; Gulianello, M.; Conway, C.M.; Li, Y.-W.; Pieschl, R.; Tian, Y.; Hong, Y.; Bristow, L.; Albright, C.F.; Hamman, B.; Allen, J.; Lippy, J.; Nara, S.; Pattipati, S.N.; Dandapani, K.; Dokania, M.; Vattikundala, P.; Sharma, V.; Elavazhagan, S.; Verma, M.K.; Lal Das, M.; Wagh, S.; Saminathan, H.; Holenarsipur, V.K.; Kumar, A.; Rao, A.; Putlur, S.P.; Sarvasiddhi, S.K.; Shankar, G.; Louis, J.V.; Ramarao, M.; Balakrishnan, A.; Johnson, B.M.; Santone, K.S.; Thalody, G.; Denton, R.
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 24 March 2022, 65(6):4534-4564)
Academic Journal
Regueiro-Ren, A.; Swidorski, J.J.; Liu, Z.; Chen, Y.; Sin, N.; Sit, S.-Y.; Chen, J.; Venables, B.L.; Easter, J.; Meanwell, N.A.; Zhu, J.; Nowicka-Sans, B.; Protack, T.; Lin, Z.; Terry, B.; Samanta, H.; Zhang, S.; Li, Z.; Cockett, M.I.; Krystal, M.; Dicker, I.B.; Beno, B.R.; Arora, V.; Huang, X.S.; Rahematpura, S.; Parker, D.D.; Haskell, R.; Santone, K.S.; Jenkins, S.; Hanumegowda, U.
In: Journal of Medicinal Chemistry . (Journal of Medicinal Chemistry, 23 August 2018, 61(16):7289-7313)
Academic Journal
Hill, M.D.; Fang, H.; Brown, J.M.; Molski, T.; Easton, A.; Han, X.; Miller, R.; Hill-Drzewi, M.; Gallagher, L.; Matchett, M.; Gulianello, M.; Balakrishnan, A.; Bertekap, R.L.; Santone, K.S.; Whiterock, V.J.; Zhuo, X.; Bronson, J.J.; Macor, J.E.; Degnan, A.P.
In: ACS Medicinal Chemistry Letters . (ACS Medicinal Chemistry Letters, 8 December 2016, 7(12):1082-1086)
Academic Journal
Kostich, W.; Li, Y.-W.; Feng, J.; Easton, A.; Bourin, C.; Gulianello, M.; Molski, T.; Brown, J.M.; Lewis, M.; Huang, Y.; Lu, Y.; Pieschl, R.; Zaczek, R.; Westphal, R.; Kiss, L.; Bristow, L.; Conway, C.M.; Albright, C.F.; Dzierba, C.; Bronson, J.; Macor, J.E.; Balakrishnan, A.; Grace, J.E.; Lentz, K.A.; Santone, K.S.; Denton, R.; O'malley, K.; Lippy, J.; Naidu, S.; Dandapani, K.; Louis, J.V.; Dokania, M.; Elavazhagan, S.; Vattikundala, P.; Sharma, V.; Das, M.L.; Shankar, G.; Kumar, A.; Holenarsipur, V.K.; Mandlekar, S.; Vikramadithyan, R.K.; Nara, S.J.; Swaffield, J.; Hamman, .B.D.; Baker, K.; Allen, J.; Savelieva, K.; Nouraldeen, A.; Lanthorn, T.H.; Ye, G.; Wilson, A.; Zambrowicz, B.; Bi, Y.; Main, A.; Carson, K.
In: Journal of Pharmacology and Experimental Therapeutics . (Journal of Pharmacology and Experimental Therapeutics, September 2016, 358(3):371-386)
Academic Journal
Regueiro-Ren, A.; Liu, Z.; Chen, Y.; Sin, N.; Sit, S.-Y.; Swidorski, J.J.; Chen, J.; Venables, B.L.; Meanwell, N.A.; Zhu, J.; Nowicka-Sans, B.; Protack, T.; Lin, Z.; Terry, B.; Samanta, H.; Zhang, S.; Li, Z.; Cockett, M.I.; Krystal, M.; Dicker, I.B.; Beno, B.R.; Huang, X.S.; Rahematpura, S.; Parker, D.D.; Haskell, R.; Jenkins, S.; Santone, K.S.; Hanumegowda, U.
In: ACS Medicinal Chemistry Letters . (ACS Medicinal Chemistry Letters, 9 June 2016, 7(6):568-572)
Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5
Academic Journal
Yang, F.; Snyder, L.B.; Balakrishnan, A.; Brown, J.M.; Sivarao, D.V.; Easton, A.; Fernandes, A.; Gulianello, M.; Hanumegowda, U.M.; Huang, H.; Huang, Y.; Jones, K.M.; Li, Y.-W.; Matchett, M.; Mattson, G.; Miller, R.; Santone, K.S.; Senapati, A.; Shields, E.E.; Simutis, F.J.; Westphal, R.; Whiterock, V.J.; Bronson, J.J.; MacOr, J.E.; Degnan, A.P.
In: ACS Medicinal Chemistry Letters . (ACS Medicinal Chemistry Letters, 10 March 2016, 7(3):289-293)
Academic Journal
Degnan, A.P.; Maxwell, D.; Balakrishnan, A.; Brown, J.M.; Easton, A.; Gulianello, M.; Hanumegowda, U.; Hill-Drzewi, M.; Miller, R.; Santone, K.S.; Senapati, A.; Shields, E.E.; Sivarao, D.V.; Westphal, R.; Whiterock, V.J.; Zhuo, X.; Bronson, J.J.; Macor, J.E.
In: Bioorganic and Medicinal Chemistry Letters . (Bioorganic and Medicinal Chemistry Letters, 2016, 26(24):5871-5876)
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[AR] Santone, K.S.
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